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Preparation of Oxysterols by C-H Oxidation of Dibromocholestane with Ru(Bpga) Catalyst.

Molecules (Basel, Switzerland)

Fujii Y, Yoritate M, Makino K, Igawa K, Takeda D, Doiuchi D, Tomooka K, Uchida T, Hirai G.
PMID: 35011456
Molecules. 2021 Dec 30;27(1). doi: 10.3390/molecules27010225.

Seven mono- and dihydroxycholesterols were prepared by direct C-H oxidation of the cholestane skeleton with a recently developed Ru(Bpga) catalyst (Ru(Bpga) = [RuCl (bpga) (PPh

Cite
Fujii Y, Yoritate M, Makino K, et al. Preparation of Oxysterols by C-H Oxidation of Dibromocholestane with Ru(Bpga) Catalyst. Molecules. 2021;27(1)doi: 10.3390/molecules27010225.
Fujii, Y., Yoritate, M., Makino, K., Igawa, K., Takeda, D., Doiuchi, D., Tomooka, K., Uchida, T., & Hirai, G. (2021). Preparation of Oxysterols by C-H Oxidation of Dibromocholestane with Ru(Bpga) Catalyst. Molecules (Basel, Switzerland), 27(1), . https://doi.org/10.3390/molecules27010225
Fujii, Yui, et al. "Preparation of Oxysterols by C-H Oxidation of Dibromocholestane with Ru(Bpga) Catalyst." Molecules (Basel, Switzerland) vol. 27,1 (2021). doi: https://doi.org/10.3390/molecules27010225
Fujii Y, Yoritate M, Makino K, Igawa K, Takeda D, Doiuchi D, Tomooka K, Uchida T, Hirai G. Preparation of Oxysterols by C-H Oxidation of Dibromocholestane with Ru(Bpga) Catalyst. Molecules. 2021 Dec 30;27(1). doi: 10.3390/molecules27010225. PMID: 35011456; PMCID: PMC8746986.
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Optimization of TAM16, a Benzofuran That Inhibits the Thioesterase Activity of Pks13; Evaluation toward a Preclinical Candidate for a Novel Antituberculosis Clinical Target.

Journal of medicinal chemistry

Wilson C, Ray P, Zuccotto F, Hernandez J, Aggarwal A, Mackenzie C, Caldwell N, Taylor M, Huggett M, Mathieson M, Murugesan D, Smith A, Davis S, Cocco M, Parai MK, Acharya A, Tamaki F, Scullion P, Epemolu O, Riley J, Stojanovski L, Lopez-Román EM, Torres-Gómez PA, Toledo AM, Guijarro-Lopez L, Camino I, Engelhart CA, Schnappinger D, Massoudi LM, Lenaerts A, Robertson GT, Walpole C, Matthews D, Floyd D, Sacchettini JC, Read KD, Encinas L, Bates RH, Green SR, Wyatt PG.
PMID: 34910486
J Med Chem. 2022 Jan 13;65(1):409-423. doi: 10.1021/acs.jmedchem.1c01586. Epub 2021 Dec 15.

With increasing drug resistance in tuberculosis (TB) patient populations, there is an urgent need for new drugs. Ideally, new agents should work through novel targets so that they are unencumbered by preexisting clinical resistance to current treatments. Benzofuran

Cite
Wilson C, Ray P, Zuccotto F, et al. Optimization of TAM16, a Benzofuran That Inhibits the Thioesterase Activity of Pks13; Evaluation toward a Preclinical Candidate for a Novel Antituberculosis Clinical Target. J Med Chem. 2021;65(1):409-423doi: 10.1021/acs.jmedchem.1c01586.
Wilson, C., Ray, P., Zuccotto, F., Hernandez, J., Aggarwal, A., Mackenzie, C., Caldwell, N., Taylor, M., Huggett, M., Mathieson, M., Murugesan, D., Smith, A., Davis, S., Cocco, M., Parai, M. K., Acharya, A., Tamaki, F., Scullion, P., Epemolu, O., Riley, J., Stojanovski, L., Lopez-Román, E. M., Torres-Gómez, P. A., Toledo, A. M., Guijarro-Lopez, L., Camino, I., Engelhart, C. A., Schnappinger, D., Massoudi, L. M., Lenaerts, A., Robertson, G. T., Walpole, C., Matthews, D., Floyd, D., Sacchettini, J. C., Read, K. D., Encinas, L., Bates, R. H., Green, S. R., & Wyatt, P. G. (2022). Optimization of TAM16, a Benzofuran That Inhibits the Thioesterase Activity of Pks13; Evaluation toward a Preclinical Candidate for a Novel Antituberculosis Clinical Target. Journal of medicinal chemistry, 65(1), 409-423. https://doi.org/10.1021/acs.jmedchem.1c01586
Wilson, Caroline, et al. "Optimization of TAM16, a Benzofuran That Inhibits the Thioesterase Activity of Pks13; Evaluation toward a Preclinical Candidate for a Novel Antituberculosis Clinical Target." Journal of medicinal chemistry vol. 65,1 (2022): 409-423. doi: https://doi.org/10.1021/acs.jmedchem.1c01586
Wilson C, Ray P, Zuccotto F, Hernandez J, Aggarwal A, Mackenzie C, Caldwell N, Taylor M, Huggett M, Mathieson M, Murugesan D, Smith A, Davis S, Cocco M, Parai MK, Acharya A, Tamaki F, Scullion P, Epemolu O, Riley J, Stojanovski L, Lopez-Román EM, Torres-Gómez PA, Toledo AM, Guijarro-Lopez L, Camino I, Engelhart CA, Schnappinger D, Massoudi LM, Lenaerts A, Robertson GT, Walpole C, Matthews D, Floyd D, Sacchettini JC, Read KD, Encinas L, Bates RH, Green SR, Wyatt PG. Optimization of TAM16, a Benzofuran That Inhibits the Thioesterase Activity of Pks13; Evaluation toward a Preclinical Candidate for a Novel Antituberculosis Clinical Target. J Med Chem. 2022 Jan 13;65(1):409-423. doi: 10.1021/acs.jmedchem.1c01586. Epub 2021 Dec 15. PMID: 34910486.
Copy Download .nbib Format: NLM
Showing 1225 to 1226 of 1226 entries