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Crystal structures of two (.

Acta crystallographica. Section E, Crystallographic communications

Galushchinskiy A, Slepukhin P, Obydennov K.
PMID: 29250401
Acta Crystallogr E Crystallogr Commun. 2017 Nov 10;73:1850-1854. doi: 10.1107/S2056989017016061. eCollection 2017 Dec 01.

The crystal structures of two (oxo-thia-zolidin-2-yl-idene)acetamides, namely (

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Galushchinskiy A, Slepukhin P, Obydennov K. Crystal structures of two (. Acta Crystallogr E Crystallogr Commun. 2017;73:1850-1854doi: 10.1107/S2056989017016061.
Galushchinskiy, A., Slepukhin, P., & Obydennov, K. (2017). Crystal structures of two (. Acta crystallographica. Section E, Crystallographic communications, 731850-1854. https://doi.org/10.1107/S2056989017016061
Galushchinskiy, Aleksei, et al. "Crystal structures of two (." Acta crystallographica. Section E, Crystallographic communications vol. 73 (2017): 1850-1854. doi: https://doi.org/10.1107/S2056989017016061
Galushchinskiy A, Slepukhin P, Obydennov K. Crystal structures of two (. Acta Crystallogr E Crystallogr Commun. 2017 Nov 10;73:1850-1854. doi: 10.1107/S2056989017016061. eCollection 2017 Dec 01. PMID: 29250401; PMCID: PMC5730238.
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Palladium-Catalyzed [3 + 2]-C-C/N-C Bond-Forming Annulation.

Organic letters

Liu Y, Mao Z, Pradal A, Huang PQ, Oble J, Poli G.
PMID: 29897775
Org Lett. 2018 Jul 06;20(13):4057-4061. doi: 10.1021/acs.orglett.8b01616. Epub 2018 Jun 13.

The synthesis of bi- and tricyclic structures incorporating pyrrolidone rings is disclosed, starting from resonance-stabilized acetamides and cyclic α,β-unsaturated-γ-oxycarbonyl derivatives. This process involves an intermolecular Tsuji-Trost allylation/intramolecular nitrogen 1,4-addition sequence. Crucial for the success of this bis-nucleophile/bis-electrophile [3 +...

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Liu Y, Mao Z, Pradal A, et al. Palladium-Catalyzed [3 + 2]-C-C/N-C Bond-Forming Annulation. Org Lett. 2018;20(13):4057-4061doi: 10.1021/acs.orglett.8b01616.
Liu, Y., Mao, Z., Pradal, A., Huang, P. Q., Oble, J., & Poli, G. (2018). Palladium-Catalyzed [3 + 2]-C-C/N-C Bond-Forming Annulation. Organic letters, 20(13), 4057-4061. https://doi.org/10.1021/acs.orglett.8b01616
Liu, Yang, et al. "Palladium-Catalyzed [3 + 2]-C-C/N-C Bond-Forming Annulation." Organic letters vol. 20,13 (2018): 4057-4061. doi: https://doi.org/10.1021/acs.orglett.8b01616
Liu Y, Mao Z, Pradal A, Huang PQ, Oble J, Poli G. Palladium-Catalyzed [3 + 2]-C-C/N-C Bond-Forming Annulation. Org Lett. 2018 Jul 06;20(13):4057-4061. doi: 10.1021/acs.orglett.8b01616. Epub 2018 Jun 13. PMID: 29897775.
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Visible-Light-Promoted Oxo-difluoroalkylation of Alkenes with DMSO as the Oxidant.

The Journal of organic chemistry

Xia ZH, Gao ZH, Dai L, Ye S.
PMID: 31083945
J Org Chem. 2019 Jun 07;84(11):7388-7394. doi: 10.1021/acs.joc.9b01077. Epub 2019 May 23.

Visible-light-promoted oxo-difluoroalkylation (acetylation and acetamidation) of alkenes with dimethyl sulfoxide as both the solvent and the oxidant was developed, affording the corresponding α,α-difluoro-γ-ketoacetates and acetamides in modest yields. Both terminal and internal alkenes worked well for the reaction. This...

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Xia ZH, Gao ZH, Dai L, et al. Visible-Light-Promoted Oxo-difluoroalkylation of Alkenes with DMSO as the Oxidant. J Org Chem. 2019;84(11):7388-7394doi: 10.1021/acs.joc.9b01077.
Xia, Z. H., Gao, Z. H., Dai, L., & Ye, S. (2019). Visible-Light-Promoted Oxo-difluoroalkylation of Alkenes with DMSO as the Oxidant. The Journal of organic chemistry, 84(11), 7388-7394. https://doi.org/10.1021/acs.joc.9b01077
Xia, Zi-Hao, et al. "Visible-Light-Promoted Oxo-difluoroalkylation of Alkenes with DMSO as the Oxidant." The Journal of organic chemistry vol. 84,11 (2019): 7388-7394. doi: https://doi.org/10.1021/acs.joc.9b01077
Xia ZH, Gao ZH, Dai L, Ye S. Visible-Light-Promoted Oxo-difluoroalkylation of Alkenes with DMSO as the Oxidant. J Org Chem. 2019 Jun 07;84(11):7388-7394. doi: 10.1021/acs.joc.9b01077. Epub 2019 May 23. PMID: 31083945.
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Design, Synthesis, and Biological Evaluation of Novel Fluorescent Probes Targeting the 18-kDa Translocator Protein.

ChemMedChem

Wongso H, Yamasaki T, Kumata K, Ono M, Higuchi M, Zhang MR, Fulham MJ, Katsifis A, Keller PA.
PMID: 33631047
ChemMedChem. 2021 Jun 17;16(12):1902-1916. doi: 10.1002/cmdc.202000984. Epub 2021 Mar 24.

A series of fluorescent probes from the 6-chloro-2-phenylimidazo[1,2-a]pyridine-3-yl acetamides ligands featuring the 7-nitro-2-oxa-1,3-diazol-4-yl (NBD) moiety has been synthesized and biologically evaluated for their fluorescence properties and for their binding affinity to the 18-kDa translocator protein (TSPO). Spectroscopic studies including...

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Wongso H, Yamasaki T, Kumata K, et al. Design, Synthesis, and Biological Evaluation of Novel Fluorescent Probes Targeting the 18-kDa Translocator Protein. ChemMedChem. 2021;16(12):1902-1916doi: 10.1002/cmdc.202000984.
Wongso, H., Yamasaki, T., Kumata, K., Ono, M., Higuchi, M., Zhang, M. R., Fulham, M. J., Katsifis, A., & Keller, P. A. (2021). Design, Synthesis, and Biological Evaluation of Novel Fluorescent Probes Targeting the 18-kDa Translocator Protein. ChemMedChem, 16(12), 1902-1916. https://doi.org/10.1002/cmdc.202000984
Wongso, Hendris, et al. "Design, Synthesis, and Biological Evaluation of Novel Fluorescent Probes Targeting the 18-kDa Translocator Protein." ChemMedChem vol. 16,12 (2021): 1902-1916. doi: https://doi.org/10.1002/cmdc.202000984
Wongso H, Yamasaki T, Kumata K, Ono M, Higuchi M, Zhang MR, Fulham MJ, Katsifis A, Keller PA. Design, Synthesis, and Biological Evaluation of Novel Fluorescent Probes Targeting the 18-kDa Translocator Protein. ChemMedChem. 2021 Jun 17;16(12):1902-1916. doi: 10.1002/cmdc.202000984. Epub 2021 Mar 24. PMID: 33631047.
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Silicon-Mediated Coupling of Carbon Monoxide, Ammonia, and Primary Amines to Form Acetamides.

Angewandte Chemie (International ed. in English)

Luecke MP, Kostenko A, Wang Y, Yao S, Driess M.
PMID: 31157488
Angew Chem Int Ed Engl. 2019 Sep 09;58(37):12940-12944. doi: 10.1002/anie.201904361. Epub 2019 Jul 08.

For the first time, a direct transformation of CO, NH

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Luecke MP, Kostenko A, Wang Y, et al. Silicon-Mediated Coupling of Carbon Monoxide, Ammonia, and Primary Amines to Form Acetamides. Angew Chem Int Ed Engl. 2019;58(37):12940-12944doi: 10.1002/anie.201904361.
Luecke, M. P., Kostenko, A., Wang, Y., Yao, S., & Driess, M. (2019). Silicon-Mediated Coupling of Carbon Monoxide, Ammonia, and Primary Amines to Form Acetamides. Angewandte Chemie (International ed. in English), 58(37), 12940-12944. https://doi.org/10.1002/anie.201904361
Luecke, Marcel-Philip, et al. "Silicon-Mediated Coupling of Carbon Monoxide, Ammonia, and Primary Amines to Form Acetamides." Angewandte Chemie (International ed. in English) vol. 58,37 (2019): 12940-12944. doi: https://doi.org/10.1002/anie.201904361
Luecke MP, Kostenko A, Wang Y, Yao S, Driess M. Silicon-Mediated Coupling of Carbon Monoxide, Ammonia, and Primary Amines to Form Acetamides. Angew Chem Int Ed Engl. 2019 Sep 09;58(37):12940-12944. doi: 10.1002/anie.201904361. Epub 2019 Jul 08. PMID: 31157488.
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Mycobacterium enoyl acyl carrier protein reductase (InhA): A key target for antitubercular drug discovery.

Bioorganic chemistry

Prasad MS, Bhole RP, Khedekar PB, Chikhale RV.
PMID: 34392175
Bioorg Chem. 2021 Oct;115:105242. doi: 10.1016/j.bioorg.2021.105242. Epub 2021 Aug 08.

Enoyl acyl carrier protein reductase (InhA) is a key enzyme involved in fatty acid synthesis mainly mycolic acid biosynthesis that is a part of NADH dependent acyl carrier protein reductase family. The aim of the present literature is to...

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Prasad MS, Bhole RP, Khedekar PB, et al. Mycobacterium enoyl acyl carrier protein reductase (InhA): A key target for antitubercular drug discovery. Bioorg Chem. 2021;115:105242doi: 10.1016/j.bioorg.2021.105242.
Prasad, M. S., Bhole, R. P., Khedekar, P. B., & Chikhale, R. V. (2021). Mycobacterium enoyl acyl carrier protein reductase (InhA): A key target for antitubercular drug discovery. Bioorganic chemistry, 115105242. https://doi.org/10.1016/j.bioorg.2021.105242
Prasad, Mayuri S, et al. "Mycobacterium enoyl acyl carrier protein reductase (InhA): A key target for antitubercular drug discovery." Bioorganic chemistry vol. 115 (2021): 105242. doi: https://doi.org/10.1016/j.bioorg.2021.105242
Prasad MS, Bhole RP, Khedekar PB, Chikhale RV. Mycobacterium enoyl acyl carrier protein reductase (InhA): A key target for antitubercular drug discovery. Bioorg Chem. 2021 Oct;115:105242. doi: 10.1016/j.bioorg.2021.105242. Epub 2021 Aug 08. PMID: 34392175.
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Photochemical C-F Activation Enables Defluorinative Alkylation of Trifluoroacetates and -Acetamides.

Journal of the American Chemical Society

Campbell MW, Polites VC, Patel S, Lipson JE, Majhi J, Molander GA.
PMID: 34793157
J Am Chem Soc. 2021 Dec 01;143(47):19648-19654. doi: 10.1021/jacs.1c11059. Epub 2021 Nov 18.

The installation of

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Campbell MW, Polites VC, Patel S, et al. Photochemical C-F Activation Enables Defluorinative Alkylation of Trifluoroacetates and -Acetamides. J Am Chem Soc. 2021;143(47):19648-19654doi: 10.1021/jacs.1c11059.
Campbell, M. W., Polites, V. C., Patel, S., Lipson, J. E., Majhi, J., & Molander, G. A. (2021). Photochemical C-F Activation Enables Defluorinative Alkylation of Trifluoroacetates and -Acetamides. Journal of the American Chemical Society, 143(47), 19648-19654. https://doi.org/10.1021/jacs.1c11059
Campbell, Mark W, et al. "Photochemical C-F Activation Enables Defluorinative Alkylation of Trifluoroacetates and -Acetamides." Journal of the American Chemical Society vol. 143,47 (2021): 19648-19654. doi: https://doi.org/10.1021/jacs.1c11059
Campbell MW, Polites VC, Patel S, Lipson JE, Majhi J, Molander GA. Photochemical C-F Activation Enables Defluorinative Alkylation of Trifluoroacetates and -Acetamides. J Am Chem Soc. 2021 Dec 01;143(47):19648-19654. doi: 10.1021/jacs.1c11059. Epub 2021 Nov 18. PMID: 34793157.
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Design, Synthesis and Biological Evaluation of a Novel Series of Thiadiazole- Based Anticancer Agents as Potent Angiogenesis Inhibitors.

Anti-cancer agents in medicinal chemistry

Altuğ-Tasa B, Kaya-Çavuşoğlu B, Koparal AT, Turan G, Koparal AS, Kaplancıklı ZA.
PMID: 33390125
Anticancer Agents Med Chem. 2021;21(15):2041-2049. doi: 10.2174/1871520621666201231143535.

BACKGROUND: Thiadiazole has attracted a great deal of interest as a versatile heterocycle for the discovery and development of potent anticancer agents. Thiadiazole derivatives exert potent antitumor activity against a variety of human cancer cell lines through various mechanisms.OBJECTIVE:...

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Altuğ-Tasa B, Kaya-Çavuşoğlu B, Koparal AT, et al. Design, Synthesis and Biological Evaluation of a Novel Series of Thiadiazole- Based Anticancer Agents as Potent Angiogenesis Inhibitors. Anticancer Agents Med Chem. 2021;21(15):2041-2049doi: 10.2174/1871520621666201231143535.
Altuğ-Tasa, B., Kaya-Çavuşoğlu, B., Koparal, A. T., Turan, G., Koparal, A. S., & Kaplancıklı, Z. A. (2021). Design, Synthesis and Biological Evaluation of a Novel Series of Thiadiazole- Based Anticancer Agents as Potent Angiogenesis Inhibitors. Anti-cancer agents in medicinal chemistry, 21(15), 2041-2049. https://doi.org/10.2174/1871520621666201231143535
Altuğ-Tasa, Burcugül, et al. "Design, Synthesis and Biological Evaluation of a Novel Series of Thiadiazole- Based Anticancer Agents as Potent Angiogenesis Inhibitors." Anti-cancer agents in medicinal chemistry vol. 21,15 (2021): 2041-2049. doi: https://doi.org/10.2174/1871520621666201231143535
Altuğ-Tasa B, Kaya-Çavuşoğlu B, Koparal AT, Turan G, Koparal AS, Kaplancıklı ZA. Design, Synthesis and Biological Evaluation of a Novel Series of Thiadiazole- Based Anticancer Agents as Potent Angiogenesis Inhibitors. Anticancer Agents Med Chem. 2021;21(15):2041-2049. doi: 10.2174/1871520621666201231143535. PMID: 33390125.
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Correction to "Indole-3-acetamides: As Potential Antihyperglycemic and Antioxidant Agents; Synthesis, .

ACS omega

Kanwal, Khan KM, Chigurupati S, Ali F, Younus M, Aldubayan M, Wadood A, Khan H, Taha M, Perveen S.
PMID: 35036820
ACS Omega. 2021 Dec 27;7(1):1541. doi: 10.1021/acsomega.1c06978. eCollection 2022 Jan 11.

[This corrects the article DOI: 10.1021/acsomega.0c05581.].

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Kanwal, Khan KM, Chigurupati S, et al. Correction to "Indole-3-acetamides: As Potential Antihyperglycemic and Antioxidant Agents; Synthesis, . ACS Omega. 2021;7(1):1541doi: 10.1021/acsomega.1c06978.
Kanwal, Khan, K. M., Chigurupati, S., Ali, F., Younus, M., Aldubayan, M., Wadood, A., Khan, H., Taha, M., & Perveen, S. (2022). Correction to "Indole-3-acetamides: As Potential Antihyperglycemic and Antioxidant Agents; Synthesis, . ACS omega, 7(1), 1541. https://doi.org/10.1021/acsomega.1c06978
Kanwal, et al. "Correction to "Indole-3-acetamides: As Potential Antihyperglycemic and Antioxidant Agents; Synthesis, ." ACS omega vol. 7,1 (2022): 1541. doi: https://doi.org/10.1021/acsomega.1c06978
Kanwal, Khan KM, Chigurupati S, Ali F, Younus M, Aldubayan M, Wadood A, Khan H, Taha M, Perveen S. Correction to "Indole-3-acetamides: As Potential Antihyperglycemic and Antioxidant Agents; Synthesis, . ACS Omega. 2021 Dec 27;7(1):1541. doi: 10.1021/acsomega.1c06978. eCollection 2022 Jan 11. PMID: 35036820; PMCID: PMC8756592.
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Anti-melanogenesis and anti-tyrosinase properties of aryl-substituted acetamides of phenoxy methyl triazole conjugated with thiosemicarbazide: Design, synthesis and biological evaluations.

Bioorganic chemistry

Hosseinpoor H, Moghadam Farid S, Iraji A, Askari S, Edraki N, Hosseini S, Jamshidzadeh A, Larijani B, Attarroshan M, Pirhadi S, Mahdavi M, Khoshneviszadeh M.
PMID: 34140181
Bioorg Chem. 2021 Sep;114:104979. doi: 10.1016/j.bioorg.2021.104979. Epub 2021 May 11.

A series of aryl phenoxy methyl triazole conjugated with thiosemicarbazides were designed, synthesized, and evaluated for their tyrosinase inhibitory activities in the presence of l-dopa and l-tyrosine as substrates. All the compounds showed tyrosinase inhibition in the sub-micromolar concentration....

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Hosseinpoor H, Moghadam Farid S, Iraji A, et al. Anti-melanogenesis and anti-tyrosinase properties of aryl-substituted acetamides of phenoxy methyl triazole conjugated with thiosemicarbazide: Design, synthesis and biological evaluations. Bioorg Chem. 2021;114:104979doi: 10.1016/j.bioorg.2021.104979.
Hosseinpoor, H., Moghadam Farid, S., Iraji, A., Askari, S., Edraki, N., Hosseini, S., Jamshidzadeh, A., Larijani, B., Attarroshan, M., Pirhadi, S., Mahdavi, M., & Khoshneviszadeh, M. (2021). Anti-melanogenesis and anti-tyrosinase properties of aryl-substituted acetamides of phenoxy methyl triazole conjugated with thiosemicarbazide: Design, synthesis and biological evaluations. Bioorganic chemistry, 114104979. https://doi.org/10.1016/j.bioorg.2021.104979
Hosseinpoor, Hona, et al. "Anti-melanogenesis and anti-tyrosinase properties of aryl-substituted acetamides of phenoxy methyl triazole conjugated with thiosemicarbazide: Design, synthesis and biological evaluations." Bioorganic chemistry vol. 114 (2021): 104979. doi: https://doi.org/10.1016/j.bioorg.2021.104979
Hosseinpoor H, Moghadam Farid S, Iraji A, Askari S, Edraki N, Hosseini S, Jamshidzadeh A, Larijani B, Attarroshan M, Pirhadi S, Mahdavi M, Khoshneviszadeh M. Anti-melanogenesis and anti-tyrosinase properties of aryl-substituted acetamides of phenoxy methyl triazole conjugated with thiosemicarbazide: Design, synthesis and biological evaluations. Bioorg Chem. 2021 Sep;114:104979. doi: 10.1016/j.bioorg.2021.104979. Epub 2021 May 11. PMID: 34140181.
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Kinetic Study of the Reaction of the Phthalimide-N-oxyl Radical with Amides: Structural and Medium Effects on the Hydrogen Atom Transfer Reactivity and Selectivity.

The Journal of organic chemistry

Bietti M, Forcina V, Lanzalunga O, Lapi A, Martin T, Mazzonna M, Salamone M.
PMID: 27934460
J Org Chem. 2016 Dec 02;81(23):11924-11931. doi: 10.1021/acs.joc.6b02482. Epub 2016 Nov 18.

A kinetic study of the hydrogen atom transfer (HAT) reactions from a series of secondary N-(4-X-benzyl)acetamides and tertiary amides to the phthalimide-N-oxyl radical (PINO) has been carried out. The results indicate that HAT is strongly influenced by structural and...

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Bietti M, Forcina V, Lanzalunga O, et al. Kinetic Study of the Reaction of the Phthalimide-N-oxyl Radical with Amides: Structural and Medium Effects on the Hydrogen Atom Transfer Reactivity and Selectivity. J Org Chem. 2016;81(23):11924-11931doi: 10.1021/acs.joc.6b02482.
Bietti, M., Forcina, V., Lanzalunga, O., Lapi, A., Martin, T., Mazzonna, M., & Salamone, M. (2016). Kinetic Study of the Reaction of the Phthalimide-N-oxyl Radical with Amides: Structural and Medium Effects on the Hydrogen Atom Transfer Reactivity and Selectivity. The Journal of organic chemistry, 81(23), 11924-11931. https://doi.org/10.1021/acs.joc.6b02482
Bietti, Massimo, et al. "Kinetic Study of the Reaction of the Phthalimide-N-oxyl Radical with Amides: Structural and Medium Effects on the Hydrogen Atom Transfer Reactivity and Selectivity." The Journal of organic chemistry vol. 81,23 (2016): 11924-11931. doi: https://doi.org/10.1021/acs.joc.6b02482
Bietti M, Forcina V, Lanzalunga O, Lapi A, Martin T, Mazzonna M, Salamone M. Kinetic Study of the Reaction of the Phthalimide-N-oxyl Radical with Amides: Structural and Medium Effects on the Hydrogen Atom Transfer Reactivity and Selectivity. J Org Chem. 2016 Dec 02;81(23):11924-11931. doi: 10.1021/acs.joc.6b02482. Epub 2016 Nov 18. PMID: 27934460.
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Base-controlled [3+3] cycloaddition of isoquinoline N-oxides with azaoxyallyl cations.

Chemical communications (Cambridge, England)

An Y, Xia H, Wu J.
PMID: 27484327
Chem Commun (Camb). 2016 Aug 16;52(68):10415-8. doi: 10.1039/c6cc03650c.

A base-controlled [3+3] cycloaddition reaction of isoquinoline N-oxides with azaoxyallyl cations is developed. 1,11b-dihydro-[1,2,4]oxadiazino[3,2-a]isoquinolin-2(3H)-ones are obtained when isoquinoline N-oxides are treated with α-halohydroxamates in the presence of sodium carbonate, while 2-(isoquinolin-1-yloxy)acetamides are unexpectedly produced when the base is changed...

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An Y, Xia H, Wu J. Base-controlled [3+3] cycloaddition of isoquinoline N-oxides with azaoxyallyl cations. Chem Commun (Camb). 2016;52(68):10415-8doi: 10.1039/c6cc03650c.
An, Y., Xia, H., & Wu, J. (2016). Base-controlled [3+3] cycloaddition of isoquinoline N-oxides with azaoxyallyl cations. Chemical communications (Cambridge, England), 52(68), 10415-8. https://doi.org/10.1039/c6cc03650c
An, Yuanyuan, et al. "Base-controlled [3+3] cycloaddition of isoquinoline N-oxides with azaoxyallyl cations." Chemical communications (Cambridge, England) vol. 52,68 (2016): 10415-8. doi: https://doi.org/10.1039/c6cc03650c
An Y, Xia H, Wu J. Base-controlled [3+3] cycloaddition of isoquinoline N-oxides with azaoxyallyl cations. Chem Commun (Camb). 2016 Aug 16;52(68):10415-8. doi: 10.1039/c6cc03650c. PMID: 27484327.
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