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J Med Chem. 2021 Oct 14;64(19):14377-14425. doi: 10.1021/acs.jmedchem.1c00888. Epub 2021 Sep 27.

Discovery of Novel UDP-.

Journal of medicinal chemistry

M Dominic Ryan, Alastair L Parkes, David Corbett, Anthony P Dickie, Michelle Southey, Ole A Andersen, Daniel B Stein, Olivier R Barbeau, Angelo Sanzone, Pia Thommes, John Barker, Ricky Cain, Christel Compper, Magali Dejob, Alain Dorali, Donnya Etheridge, Sian Evans, Adele Faulkner, Elise Gadouleau, Timothy Gorman, Denes Haase, Maisie Holbrow-Wilshaw, Thomas Krulle, Xianfu Li, Christopher Lumley, Barbara Mertins, Spencer Napier, Rajesh Odedra, Kostas Papadopoulos, Vasileios Roumpelakis, Kate Spear, Emily Trimby, Jennifer Williams, Michael Zahn, Anthony D Keefe, Ying Zhang, Holly T Soutter, Paolo A Centrella, Matthew A Clark, John W Cuozzo, Christoph E Dumelin, Boer Deng, Avery Hunt, Eric A Sigel, Dawn M Troast, Boudewijn L M DeJonge

Affiliations

  1. X-Biotix Therapeutics, 465 Waverly Oaks Road, Waltham, Massachusetts 02452, United States.
  2. Evotec, 114 Innovation Drive, Milton Park, Abingdon, Oxfordshire OX14 4RZ, U.K.
  3. Evotec UK, Anti-infectives, Block 23F, Alderley Park, Cheshire SK10 4TG, U.K.
  4. Evotec SE, Manfred Eigen Campus, Essener Bogen 7, 22419 Hamburg, Germany.
  5. X-Chem, 100 Beaver Street, Waltham, Massachusetts 02453, United States.

PMID: 34569791 DOI: 10.1021/acs.jmedchem.1c00888

Abstract

This study describes a novel series of UDP-

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